Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Keywords

Uncompetitive inhibitorNon-competitive inhibitionKineticsEnzyme kineticsSubstrate (aquarium)ChemistryEnzymeStereochemistryActive siteBiochemistryBiologyPhysics

Affiliated Institutions

Yale University US

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Publication Info

Year: 1973
Type: article
Volume: 22
Issue: 23
Pages: 3099-3108
Citations: 12771
Access: Closed

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APA Style

                            
                                    Yung-Chi Cheng, 
                                
                                    William H. Prusoff
                                
                            (1973). 
                            Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction. 
                            Biochemical Pharmacology
                            , 22
                            (23)
                            , 3099-3108.
                            https://doi.org/10.1016/0006-2952(73)90196-2

Identifiers

DOI: 10.1016/0006-2952(73)90196-2