Figure S4 from RTK-Dependent Inducible Degradation of Mutant PI3Kα Drives GDC-0077 (Inavolisib) Efficacy

Kyung Song; Kyle A. Edgar; Emily J. Hanan; Marc Hafner; Jason Oeh; Mark Merchant; Deepak Sampath; Michelle Nannini; Rebecca Hong; Lilian Phu; William F. Forrest; Eric Stawiski; Stephen D. Schmidt; Nicholas Endres; Jane Guan; Jeffrey J. Wallin; Jonathan Cheong; Emile G. Plise; Gail D. Lewis Phillips; Laurent Salphati; Timothy P. Heffron; Alan G. Olivero; Shiva Malek; Steven T. Staben; Donald S. Kirkpatrick; Anwesha Dey; Lori S. Friedman

doi:10.1158/2159-8290.30833958

Abstract

<p>Taselisib depletes mutant p110a protein through ubiquitin and proteasome mechanism in a dose and time dependent manner</p>

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Year: 2025
Type: article
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APA Style

                            
                                    Kyung Song, 
                                
                                    Kyle A. Edgar, 
                                
                                    Emily J. Hanan
                                
                                et al.
                            
                            (2025). 
                            Figure S4 from RTK-Dependent Inducible Degradation of Mutant PI3Kα Drives GDC-0077 (Inavolisib) Efficacy. 
                            
                            .
                            https://doi.org/10.1158/2159-8290.30833958

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DOI: 10.1158/2159-8290.30833958